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dopamine receptor D4
dopamine receptor D4
D-1 dopamine receptor changes after striatal quinolinic acid lesion
Animals / Male / dopamine receptor D4 / Dopamine Receptors / European / Rats / Pyridines / Autoradiography / Brain Chemistry / Dopamine antagonists / Corpus striatum / Rats / Pyridines / Autoradiography / Brain Chemistry / Dopamine antagonists / Corpus striatum
Dopaminergic Supersensitivity in G Protein-Coupled Receptor Kinase 6Deficient Mice
Cognitive Science / Animal Behavior / Dopamine / Mice / Animals / Cocaine / Amphetamine / dopamine receptor D4 / Neurons / Neuron / Gene Targeting / G protein / Neurosciences / Motor activity / Corpus striatum / Cocaine / Amphetamine / dopamine receptor D4 / Neurons / Neuron / Gene Targeting / G protein / Neurosciences / Motor activity / Corpus striatum
Preparation and Pharmacological Characterization of trans -2-Amino-5(6)-fluoro-6(5)-hydroxy-1-phenyl-2,3-dihydro-1 H -indenes as D 2 -like Dopamine Receptor Agonists
Organic Chemistry / Medicinal Chemistry / cyclic AMP / Animals / dopamine receptor D4 / Rats / Swine / Radioligand Assay / Medicinal / Structure activity Relationship / cyclic GMP / Rats / Swine / Radioligand Assay / Medicinal / Structure activity Relationship / cyclic GMP
Rolipram: A specific phosphodiesterase 4 inhibitor with potential antipsychotic activity
Neuroscience / Psychology / Psychopharmacology / Animal Behavior / Schizophrenia / Memory / Startle Reflex / Prepulse Inhibition / Mice / ANOVA / Animals / Male / PPI / dopamine receptor D4 / Animal Model / Haloperidol / Phosphodiesterase Inhibitors / Pde / Side Effect / EPS / Second Messengers / Effective Dose / Neurosciences / Dextroamphetamine / Acoustic Stimulation / Memory / Startle Reflex / Prepulse Inhibition / Mice / ANOVA / Animals / Male / PPI / dopamine receptor D4 / Animal Model / Haloperidol / Phosphodiesterase Inhibitors / Pde / Side Effect / EPS / Second Messengers / Effective Dose / Neurosciences / Dextroamphetamine / Acoustic Stimulation
Preparation and Pharmacological Characterization of trans -2-Amino-5(6)-fluoro-6(5)-hydroxy-1-phenyl-2,3-dihydro-1 H -indenes as D 2 -like Dopamine Receptor Agonists
Organic Chemistry / Medicinal Chemistry / cyclic AMP / Animals / dopamine receptor D4 / Rats / Swine / Radioligand Assay / Medicinal / Structure activity Relationship / cyclic GMP / Rats / Swine / Radioligand Assay / Medicinal / Structure activity Relationship / cyclic GMP
Lentiviral Overexpression of GRK6 Alleviates L-Dopa-Induced Dyskinesia in Experimental Parkinson\'s Disease
Animal Behavior / MicroRNA / Signal Transduction / Biological Sciences / Dopamine / Macaca / Humans / Endocytosis / Animals / dopamine receptor D4 / Lentivirus / Substantia nigra / Levodopa / Rats / Degeneration / Rotation / Macaca / Humans / Endocytosis / Animals / dopamine receptor D4 / Lentivirus / Substantia nigra / Levodopa / Rats / Degeneration / Rotation
Lentiviral Overexpression of GRK6 Alleviates L-Dopa-Induced Dyskinesia in Experimental Parkinson\'s Disease
Animal Behavior / MicroRNA / Signal Transduction / Biological Sciences / Dopamine / Macaca / Humans / Endocytosis / Animals / dopamine receptor D4 / Lentivirus / Substantia nigra / Levodopa / Rats / Degeneration / Rotation / Macaca / Humans / Endocytosis / Animals / dopamine receptor D4 / Lentivirus / Substantia nigra / Levodopa / Rats / Degeneration / Rotation
N-[11C]Methylspiperone PET, in contrast to [11C]raclopride, fails to detect D2 receptor occupancy by an atypical neuroleptic
Cognitive Science / Psychiatry / Schizophrenia / Kinetics / Positron Emission Tomography / Dopamine / Humans / Cerebellum / Caudate Nucleus / Vitamin D receptor / Male / dopamine receptor D4 / Steady state / Clinical Sciences / Single Photon Emission Computed Tomography / Adult / Putamen / Neurosciences / Dissociation Constant / Dopamine / Humans / Cerebellum / Caudate Nucleus / Vitamin D receptor / Male / dopamine receptor D4 / Steady state / Clinical Sciences / Single Photon Emission Computed Tomography / Adult / Putamen / Neurosciences / Dissociation Constant
Amisulpride is a preferential D3 dopamine receptor antagonist
Biological Sciences / Biological Psychiatry / dopamine receptor D4
Cariprazine (RGH-188), a potent D3/D2 dopamine receptor partial agonist, binds to dopamine D3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents
Neurochemistry / Dopamine / Mice / Blood brain barrier / Animals / Male / dopamine receptor D4 / Rats / Atypical Antipsychotics / Wistar Rats / Protein Binding / Neurosciences / Male / dopamine receptor D4 / Rats / Atypical Antipsychotics / Wistar Rats / Protein Binding / Neurosciences
Rolipram: A specific phosphodiesterase 4 inhibitor with potential antipsychotic activity
Neuroscience / Psychology / Animal Behavior / Memory / Startle Reflex / Prepulse Inhibition / Mice / Animals / Male / dopamine receptor D4 / Haloperidol / Phosphodiesterase Inhibitors / Side Effect / Second Messengers / Effective Dose / Neurosciences / Dextroamphetamine / Prepulse Inhibition / Mice / Animals / Male / dopamine receptor D4 / Haloperidol / Phosphodiesterase Inhibitors / Side Effect / Second Messengers / Effective Dose / Neurosciences / Dextroamphetamine
Preparation and Pharmacological Characterization of trans -2-Amino-5(6)-fluoro-6(5)-hydroxy-1-phenyl-2,3-dihydro-1 H -indenes as D 2 -like Dopamine Receptor Agonists
Organic Chemistry / Medicinal Chemistry / cyclic AMP / Animals / dopamine receptor D4 / Rats / Swine / Radioligand Assay / Medicinal / Structure activity Relationship / cyclic GMP / Rats / Swine / Radioligand Assay / Medicinal / Structure activity Relationship / cyclic GMP
Cariprazine (RGH-188), a potent D3/D2 dopamine receptor partial agonist, binds to dopamine D3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents
Neurochemistry / Dopamine / Mice / Blood brain barrier / Animals / Male / dopamine receptor D4 / Rats / Atypical Antipsychotics / Wistar Rats / Protein Binding / Neurosciences / Male / dopamine receptor D4 / Rats / Atypical Antipsychotics / Wistar Rats / Protein Binding / Neurosciences
Lentiviral Overexpression of GRK6 Alleviates L-Dopa-Induced Dyskinesia in Experimental Parkinson\'s Disease
Animal Behavior / MicroRNA / Signal Transduction / Biological Sciences / Dopamine / Macaca / Humans / Endocytosis / Animals / dopamine receptor D4 / Lentivirus / Substantia nigra / Levodopa / Rats / Degeneration / Rotation / Macaca / Humans / Endocytosis / Animals / dopamine receptor D4 / Lentivirus / Substantia nigra / Levodopa / Rats / Degeneration / Rotation
Pre- and postsynaptic dopaminergic activities of indolizidine and quinolizidine derivatives of 3-(3-hydroxyphenyl)-N-(n-propyl)piperidine (3-PPP). Further developments of a dopamine receptor model
Organic Chemistry / Medicinal Chemistry / Animals / Structural equation models / Male / dopamine receptor D4 / Dopamine Receptors / Rats / Medicinal / Molecular Conformation / Structure activity Relationship / Piperidines / Motor activity / dopamine receptor D4 / Dopamine Receptors / Rats / Medicinal / Molecular Conformation / Structure activity Relationship / Piperidines / Motor activity
Pre- and postsynaptic dopaminergic activities of indolizidine and quinolizidine derivatives of 3-(3-hydroxyphenyl)-N-(n-propyl)piperidine (3-PPP). Further developments of a dopamine receptor model
Organic Chemistry / Medicinal Chemistry / Animals / Structural equation models / Male / dopamine receptor D4 / Dopamine Receptors / Rats / Molecular Conformation / Structure activity Relationship / Piperidines / Motor activity / dopamine receptor D4 / Dopamine Receptors / Rats / Molecular Conformation / Structure activity Relationship / Piperidines / Motor activity
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